NUI
No nā nīnau e pili ana i kā mākou huahana a i ʻole ka papa inoa kumukūʻai, e ʻoluʻolu e waiho i kāu leka uila iā mākou a e hoʻopili mākou i loko o 24 mau hola.
NINAU ANOKūlana halihali
Hiki i ka wela maʻamau
Manaʻo i ke ʻano hoʻouna
Ma ka lewa Ma ka aina Ma ke kai
Kūlana mālama:
E mālama i kahi pōʻeleʻele, Inert ea, lumi wela
Ola ola
Ma kahi o 2 makahiki
Ka nui o ke kauoha liʻiliʻi:
1kg (kūkākūkā)
palapala hōʻoia:COA, wahi hehee, Hoʻololi kikoʻī [α]D20
E hoʻouna mākou i nā ʻikepili āu e makemake ai.Hiki iā ʻoe ke ʻike i ka ʻikepili ma mua ma ke ʻano he kuhikuhi.
No nā huahana maʻamau, hoʻouna mākou i ka ʻikepili hou ma hope o ka puka ʻana mai.
H-ME-LEU-OBZLTOS-OH;
N-ALPHA-METHYL-L-LEUCINEBENZYLESTERP-TOSYLATE;
benzyl(2S)-4-methyl-2-(methylamino)pentanoate;
N-METHYL-L-LEUCINEBENZYLESTER4-TOLUENESULFONATESALT;
N-ME-LEUCINE-OBZLP-TOSYLATE;
N-ME-LEU-OBZLP-TOSYLATE;
N-ME-LEU-OBZLTOSOH;
HN-Me-Leu-OBzl.TosOH
Hoʻohana pinepine ʻia lākou no ka hoʻopili ʻana i ka pauka.Pili ia i nā koi o nā mea kūʻai aku.No laila, e haʻi mai iā mākou i kāu koi ma mua o ka hoʻopaʻa ʻana inā loaʻa iā ʻoe nā noi kūikawā.
1kg a 25kg He paʻakikī ka paʻi waho.A he mea paʻakikī ke ʻoki a hōʻino.Hiki iā ia ke pale pono i kāu mau huahana.
ʻO HN-Me-Leu-Obzl.Tos-OH (N-Methyl-L-leucyl-O-benzyl-L-tyrosine tosylate) he hui peptide kiko'ī me nā mea hiki ke hoʻohana ʻia ma nā kahua he nui.
ʻO ka mea mua, ma ka noiʻi biochemical, hiki i ka HN-Me-Leu-Obzl.Tos-OH ke lawelawe ma ke ʻano he moleke bioactive e ʻimi i nā pilina a me nā ʻano hoʻoponopono o nā protein pili a i ʻole nā enzyme i loko o nā ʻōnaehana olaola.Eia hou, hiki ke hoʻohana ʻia ma ke ʻano he precursor no ka synthesizing ʻoi aku ka paʻakikī o nā peptides a i ʻole nā protein, e hāʻawi ana i kahi ʻike hohonu o ke ʻano a me ka hana o nā macromolecules biological.
ʻO ka lua, ma ke kahua o ka loaʻa ʻana o ka lāʻau lapaʻau, hiki i ka HN-Me-Leu-Obzl.Tos-OH ke hōʻike i ka hana pharmacological hiki ke hōʻike i nā hopena therapeutic i kekahi mau maʻi a i ʻole nā kaʻina pathological.No laila, hiki paha ke lilo i moho no nā lāʻau lapaʻau hou a i ʻole kahi precursor synthetic no nā alakaʻi lāʻau, e hāʻawi ana i nā ala hou a me nā ala no ka hoʻomohala ʻana i ka lāʻau.
Eia kekahi, ma ka ʻepekema waiwai, hiki i ka HN-Me-Leu-Obzl.Tos-OH ke paʻa i ka waiwai noi kūikawā.Hiki ke hana koʻikoʻi kona ʻano kemika a me kāna mau waiwai i ka hoʻomākaukau ʻana a i ʻole ka hoʻololi ʻana i nā mea kikoʻī, no laila e holomua ana i ka hoʻomohala ʻana i ka ʻepekema waiwai.
HD-Leu-OH | N-Me-L-Leu | N-Me-D-Leu-Obzl | H-Leu-OBzl.HCl |
HD-Leu-OBzl.Tos-OH | L-Leu-Otbu-OH |
1. No ka MOQ: Hiki iā mākou ke hoʻololi e like me kāu koi.
2. E pili ana i ka hāpana: Pono ka hāpana i ka uku hōʻailona, hiki ke lawe i ka ukana e hōʻiliʻili aiʻole hiki iāʻoe ke uku iā mākou ma mua.
3. Mold workshop, hiki ke hoʻopilikino ʻia e like me ka helu o nā hiʻohiʻona.
4. Hāʻawi mākou i ka lawelawe maikaʻi loa.Ke hana nei kekahi hui kūʻai akamai iā ʻoe.
5. E pili ana i ka hoʻololi: E ʻoluʻolu e leka uila a kamaʻilio paha iaʻu ma kou ʻoluʻolu.